
Tetracaine Base is a premium-grade, highly lipophilic ester-type local anesthetic active pharmaceutical ingredient (API) carrying CAS number 94-24-6. This high-purity crystalline compound is widely utilized across the global healthcare sector to manufacture clinical-strength topical anesthetic gels, ophthalmic solutions, and advanced nerve block configurations requiring prolonged anesthetic duration.
Exceptional lipid permeability and rapid cellular action provide a major competitive advantage in the formulation of therapeutic treatments. This active pharmaceutical ingredient works by providing the essential structural mechanisms—specifically binding to the intracellular portion of sodium channels to prevent sensory membrane depolarization—needed for effective systemic modulation. It helps manufacturers achieve potent numbing profiles in over-the-counter and prescription topical formulas without sacrificing formula stability. For instance, Tetracaine Base is frequently used as a primary ingredient in clinical-strength dermatological anesthetics. Consequently, it improves the final clinical efficacy of superficial surgical interventions and acute pain management routines. As a result, Zyntex ensures low heavy metal content and strict microbiological control for our supply, ensuring maximum safety during your manufacturing cycle.
Moreover, Zyntex supplies specialized fine crystalline powder grades for the human clinical compounding and specialty pharmaceutical industries. This compound acts as a critical structural asset, helping to enhance the direct numbing defense mechanisms of biological systems undergoing intense surface irritation or procedural discomfort exposure. It pushes the boundaries of medical science by offering a highly stable active source that does not affect the final solution’s target properties unless requested during direct cream blending or base compounding. At the same time, it serves as a crucial biomaterial matrix in the synthesis of specialized prolonged-release anesthetic matrices and fine chemical drug intermediates. In short, our product serves as a dependable “structural matrix.” It supports both the vitality of the human body and the precision of modern biomedical engineering.
This high-purity crystalline local anesthetic active compound is essential in these four primary sectors:
Primary active pharmaceutical source used for compounding dermal numbing creams, gels, and patches. Thus, it provides essential support for localized membrane desensitization.
Key drug ingredient utilized for preparing fast-acting anesthetic eye drops and liquid diagnostics. Undoubtedly, it is vital for enhancing immediate corneal numbing benchmarks.
Used as a professional anesthetic active for manufacturing immediate-relief dental and rhinological configurations. Consequently, it is vital for high-performance endoscopic pre-treatments.
Acts as an essential reference standard block for modern neuronal pathway mapping and industrial drug trials. Specifically, it supports rapid compounding runs and uniform molecule clarity.
| Parameter | Standard Value |
|---|---|
| Product Name | Tetracaine Base |
| Assay / Purity | 99.0% – 101.0% (Calculated on Dried Basis) |
| Appearance | White to off-white crystalline fine powder |
| Melting Point | 41 °C to 45 °C |
| Loss on Drying | ≤ 0.5% |
| CAS Number | 94-24-6 |
📝 Safety & Handling: Formulated strictly for controlled pharmaceutical manufacturing, anesthetic compounding, and clinical laboratory workflows. Tetracaine Base is an exceptionally potent active pharmaceutical drug substance with high systemic toxicity. Accidental exposure, workplace inhalation, or skin contact can induce immediate localized numbness, severe eye irritation, cardiac pathway modifications, or hypersensitivity loop reactions. Due to its remarkably low melting point parameters (41°C–45°C), it can degrade or soften under thermal stress. Therefore, store strictly in a cool, dry, dark location below 20°C, completely protected from direct sunlight fields, ambient humidity, and strong incompatible oxidizing materials in its original safety-sealed airtight containers. Avoid fine dust generation or physical contact during mass blending scales to secure laboratory personnel. Wearing full specialized protective equipment (PPE)—including chemical-resistant nitrile gloves, safety goggles, lab coats, and a certified dust respirator mask—is strictly mandatory. Always consult the Safety Data Sheet (SDS) for detailed environmental protocols.