
Dimenhydrinate is a premium-grade, high-purity antihistamine and antiemetic active pharmaceutical ingredient (API) with CAS number 523-87-5. This highly effective crystalline compound is widely utilized across the global healthcare sector to manufacture clinical-strength motion sickness tablets, motion-induced nausea liquid formulations, and advanced travel-sickness prevention solutions.
Exceptional digestibility and rapid molecular action provide a major competitive advantage in the formulation of therapeutic treatments. This active pharmaceutical ingredient works by providing the essential structural mechanisms—specifically combining diphenhydramine and 8-chlorotheophylline to block central emetic stimulation—needed for effective systemic modulation. It helps manufacturers achieve potent anti-nausea profiles in over-the-counter and prescription products without sacrificing formula stability. For instance, Dimenhydrinate is frequently used as a primary ingredient in clinical-strength motion sickness therapies. Consequently, it improves the clinical efficacy of acute vertigo and balance breakdown management routines. As a result, Zyntex ensures low heavy metal content and strict microbiological control for our supply, ensuring maximum safety during your manufacturing cycle.
Moreover, Zyntex supplies specialized fine crystalline grades for the human clinical and healthcare compounding industries. This compound acts as a critical structural asset, helping to enhance the defense mechanisms of biological systems undergoing severe inner ear hyper-reactivity exposure. It pushes the boundaries of medical science by offering a highly stable active source that does not affect the final solution’s processing parameters during direct tablet compression or wet blending. At the same time, it serves as a crucial biomaterial matrix in the synthesis of specialized combination therapies and chemical drug intermediates. In short, our product serves as a dependable “structural matrix.” It supports both the vitality of the human body and the precision of modern biomedical engineering.
This high-purity crystalline anti-nausea drug compound is essential in these four primary sectors:
Primary active pharmaceutical source used for compressing standard anti-nausea oral tablets and chewable travel caplets. Thus, it provides essential support for localized vestibular calm.
Key drug ingredient utilized for preparing stable pediatric suspensions and oral fluid formulations. Undoubtedly, it is vital for enhancing uniform dose and liquid formulation benchmarks.
Used as a specialized compounding active for manufacturing immediate relief intravenous solutions and vials. Consequently, it is vital for high-performance emergency recovery lines.
Acts as an essential reference standard block for modern H1 histaminic pathway and drug matching procedures. Specifically, it supports rapid compounding runs and uniform molecule clarity.
| Parameter | Standard Value |
|---|---|
| Product Name | Dimenhydrinate (USP / BP / EP Pharmaceutical API Grade) |
| Assay / Purity | 98.0% – 102.0% (Calculated on Dried Basis) |
| Appearance | White, crystalline, odorless powder |
| Melting Point | 102 °C to 107 °C |
| Loss on Drying | ≤ 0.5% |
| CAS Number | 523-87-5 |
📝 Safety & Handling: Formulated strictly for controlled pharmaceutical manufacturing, antiemetic compounding, and clinical laboratory workflows. Dimenhydrinate is a highly potent active antihistaminic salt derivative that can induce significant central nervous system drowsiness, sedation, mild blurred vision, or dryness of mucous membranes upon accidental inhalation or heavy exposure. Therefore, store strictly in a cool, dry location below 25°C away from direct sunlight, ambient dampness, and strong incompatible oxidizing formulations in its original tightly sealed safety containers. Prevent fine dust accumulation loops to secure chemical efficacy during mass blending steps. Wearing standard laboratory protective equipment (PPE)—including nitrile gloves, protective eyewear, and a certified dust respirator mask—is mandatory to avoid occupational exposure. Always consult the Safety Data Sheet (SDS) for detailed environmental protocols.